SCHEMBL5503174

SCHEMBL5503174

CC(=O)Nc1nc(C=Cc2ccc(OC(C)=O)cc2)c(Cc2ccc(S(C)(=O)=O)cc2)s1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 10/20 0.49
PIK3CD O00329 1/20 0.42
PIK3CA P42336 1/20 0.42
PIK3CB P42338 1/20 0.42
PIK3CG P48736 1/20 0.42
KDM4E B2RXH2 2/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
TTR P02766 1/20 0.40
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
ALDH1A1 P00352 1/20 0.38
RORC P51449 1/20 0.37
PTGS2 P35354 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4874836 0.87 AOC3 (0.49) AOC3PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL4874841 0.87 AOC3 (0.49) AOC3PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL3932528 0.87 AOC3 (0.50) AOC3PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL3936307 0.87 AOC3 (0.50) AOC3PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL6264653 0.87 AOC3 (0.50) AOC3PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL3932522 0.87 AOC3 (0.50) AOC3PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL6264646 0.87 AOC3 (0.50) AOC3PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL3939275 0.85 AOC3 (0.49) AOC3PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL3939278 0.85 AOC3 (0.49) AOC3PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL3941424 0.85 AOC3 (0.49) AOC3PIK3CDPIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786792-A2 THIAZOLE DERIVATIVES HAVING VAP-1 INHIBITORY ACTIVITY Astellas Pharma Inc. (JP) 2007-05-23 EP disclosed
WO-2006011631-A2 THIAZOLE DERIVATIVES HAVING VAP-1 INHIBITORY ACTIVITY ASTELLAS PHARMA INC. (JP) 2006-02-02 WO disclosed