SCHEMBL5503532

SCHEMBL5503532

COc1ccc2nccc(OC[C@@H]3CC[C@@H](N)CO3)c2c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 3/20 0.41
KDM4E B2RXH2 2/20 0.41
KCNH2 Q12809 2/20 0.41
HTR1A P08908 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
MET P08581 4/20 0.40
LMNA P02545 1/20 0.39
DDR2 Q16832 1/20 0.39
NCF1 P14598 1/20 0.38
MAPK1 P28482 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5507590 0.84 IRAK4 (0.41) IRAK4KCNH2
SCHEMBL3692448 0.84 KDM4E (0.46) IRAK4KDM4EKCNH2HTR1AADRA1D
SCHEMBL3692451 0.84 KDM4E (0.46) IRAK4KDM4EKCNH2HTR1AADRA1D
SCHEMBL5509173 0.84 MTNR1B (0.41) IRAK4HTR1ANCF1
SCHEMBL5503330 0.83 MTNR1B (0.43) IRAK4KDM4E
SCHEMBL5504441 0.82 KCNH2 (0.41) IRAK4KCNH2HTR1AMETLMNA
SCHEMBL4512730 0.81 KCNH2 (0.37) KCNH2
SCHEMBL5506070 0.76 MTNR1B (0.52) IRAK4
SCHEMBL591215 0.73 KDM4E (0.44) KDM4EKCNH2HTR1AADRA1DADRA1A
SCHEMBL591216 0.73 KDM4E (0.44) KDM4EKCNH2HTR1AADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799676-A2 NEW BICYCLIC ANTIBIOTICS Actelion Pharmaceuticals Ltd. (CH) 2007-06-27 EP disclosed
WO-2006032466-A2 NEW BICYCLIC ANTIBIOTICS ACTELION PHARMACEUTICALS LTD (CH) 2006-03-30 WO disclosed