SCHEMBL5503879

SCHEMBL5503879

Cc1cccc(Oc2ccc(C#N)c(Cl)c2)c1.N#Cc1ccc(Oc2cccc3ccccc23)cc1Cl

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.62
ALDH1A1 P00352 2/20 0.43
GAA P10253 1/20 0.43
SLC22A12 Q96S37 5/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
BCL2 P10415 1/20 0.39
MCL1 Q07820 1/20 0.39
PGR P06401 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4175939 0.90 AR (0.66) ARALDH1A1GAASLC22A12PGR
SCHEMBL4188869 0.86 AR (0.67) ARALDH1A1SLC22A12L3MBTL1PGR
SCHEMBL2354199 0.81 ALDH1A1 (0.62) ARALDH1A1GAAL3MBTL1
SCHEMBL9502758 0.78 ALDH1A1 (0.48) ARALDH1A1GAA
SCHEMBL4175953 0.77 AR (1.00) ARGAASLC22A12PGR
SCHEMBL8543199 0.76 AR (0.62) ARALDH1A1GAASLC22A12PGR
SCHEMBL13890551 0.75 AR (0.75) ARGAASLC22A12
SCHEMBL753907 0.75 AR (0.75) ARGAASLC22A12PGR
SCHEMBL30426714 0.75 AR (0.66) ARALDH1A1GAAL3MBTL1
SCHEMBL4184922 0.75 AR (0.65) ARALDH1A1SLC22A12PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781280-A2 ANDROGEN MODULATORS Warner-Lambert Company LLC (US) 2007-05-09 EP disclosed
WO-2006018723-A2 ANDROGEN MODULATORS WARNER-LAMBERT COMPANY LLC (US) 2006-02-23 WO disclosed