SCHEMBL5503909

SCHEMBL5503909

NS(=O)(=O)NCCC[C@@](O)(c1cccc(Cl)c1)C1CCCN(C(=O)O)C1

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
REN P00797 19/20 0.68
HTR1A P08908 1/20 0.41
DRD2 P14416 1/20 0.41
HTR2A P28223 1/20 0.41
HTR7 P34969 1/20 0.41
HTR6 P50406 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27829352 1.00 REN (0.68) RENHTR1ADRD2HTR2AHTR7
SCHEMBL1860767 0.88 REN (0.68) REN
SCHEMBL1860766 0.88 REN (0.68) REN
SCHEMBL5515427 0.86 REN (0.65) REN
SCHEMBL4752903 0.86 REN (0.53) REN
SCHEMBL5510417 0.86 REN (0.53) REN
SCHEMBL5603647 0.85 REN (0.69) REN
SCHEMBL5509846 0.85 REN (0.69) REN
SCHEMBL27689729 0.84 REN (0.70) REN
SCHEMBL27758544 0.84 REN (0.69) REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101072561-B Diaminoalkane aspartic protease inhibitors VITAE PHARMACEUTICALS INC 2011-05-11 CN disclosed
EP-1807078-A1 DIAMINOALKANE ASPARTIC PROTEASE INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2007-07-18 EP disclosed
WO-2006042150-A1 DIAMINOALKANE ASPARTIC PROTEASE INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2006-04-20 WO disclosed