SCHEMBL5504550

SCHEMBL5504550

c1cnc(C2CCNC23CC3)cn1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.34
GSK3B P49841 1/20 0.31
DYRK1A Q13627 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNA4 P43681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3464226 0.78 NISCH (0.33) NISCHCHRNB2CHRNA4
SCHEMBL5508758 0.70 CHRNB2 (0.32) CHRNB2CHRNA4
SCHEMBL9557396 0.69 HRH3 (0.44) NISCHGSK3BDYRK1A
SCHEMBL29891608 0.69 HRH3 (0.44) NISCHGSK3BDYRK1A
Hydrochloric Acid SCHEMBL20744274 0.68 HRH3 (0.43) NISCHGSK3BDYRK1A
SCHEMBL29506048 0.68 NISCH (0.30) NISCH
SCHEMBL3954850 0.67 CHEK1 (0.41) NISCHGSK3BDYRK1ACHRNB2CHRNA4
SCHEMBL29889443 0.67 CHEK1 (0.41) NISCHGSK3BDYRK1ACHRNB2CHRNA4
SCHEMBL19116619 0.67 CHEK1 (0.41) NISCHGSK3BDYRK1ACHRNB2CHRNA4
SCHEMBL8271401 0.67 CHEK1 (0.41) NISCHGSK3BDYRK1ACHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802601-A1 AZASPIROALKENE AND AZAPIROALKANE COMPOUNDS WITH NICOTINIC CHOLINERGIC RECEPTOR ACTIVITY Targacept, Inc. (US) 2007-07-04 EP claimed
WO-2006034089-A1 AZASPIROALKENE AND AZASPIROALKANE COMPOUNDS WITH NICOTINIC CHOLINERGIC RECEPTOR ACTIVITY TARGACEPT, INC. (US) 2006-03-30 WO claimed