SCHEMBL5504568

SCHEMBL5504568

CCCCCc1nc(N)co1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.37
NOS2 P35228 1/20 0.37
TLR8 Q9NR97 4/20 0.36
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
PPARA Q07869 1/20 0.35
ALDH1A1 P00352 2/20 0.34
TLR7 Q9NYK1 4/20 0.34
PI4KA P42356 1/20 0.34
PI4K2B Q8TCG2 1/20 0.34
PI4K2A Q9BTU6 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
HTR2A P28223 1/20 0.33
DHFR P00374 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2867677 0.78 KCNH2 (0.47) KCNH2NOS2S1PR1S1PR3PPARA
SCHEMBL2682119 0.78 FPR2 (0.46)
SCHEMBL27854898 0.77
SCHEMBL14764837 0.77 KCNH2 (0.37) KCNH2S1PR1S1PR3PPARAALDH1A1
SCHEMBL3663915 0.74 KCNH2 (0.39) KCNH2S1PR1S1PR3PPARAALDH1A1
SCHEMBL15448352 0.73 GCGR (0.44) KCNH2TLR8S1PR1S1PR3ALDH1A1
SCHEMBL28341385 0.72 KCNH2 (0.39) KCNH2NOS2TLR8S1PR1S1PR3
SCHEMBL5544212 0.72 KCNH2 (0.41) KCNH2NOS2S1PR1S1PR3PPARA
SCHEMBL5548022 0.70 KCNH2 (0.43) KCNH2S1PR1S1PR3PPARAALDH1A1
SCHEMBL544961 0.69 KCNH2 (0.46) KCNH2NOS2TLR8ALDH1A1TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758654-A1 USE OF C-KIT INHIBITORS FOR TREATING PLASMODIUM RELATED DISEASES AB Science (FR) 2007-03-07 EP disclosed
WO-2005102455-A1 USE OF C-KIT INHIBITORS FOR TREATING PLASMODIUM RELATED DISEASES AB SCIENCE (FR) 2005-11-03 WO disclosed