SCHEMBL5504786

SCHEMBL5504786

Nc1nc(NCC(O)C(CO)Nc2nc(N)nc3cc(-c4c(F)cccc4F)ccc23)c2ccc(-c3c(Cl)cccc3Cl)cc2n1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.37
NLRP3 Q96P20 4/20 0.36
APP P05067 2/20 0.34
CYP2D6 P10635 2/20 0.33
TLR8 Q9NR97 2/20 0.33
TLR7 Q9NYK1 1/20 0.33
MAP4K4 O95819 1/20 0.33
DRD1 P21728 1/20 0.33
HTR2A P28223 1/20 0.33
ADORA1 P30542 1/20 0.33
CDC7 O00311 1/20 0.32
NTRK1 P04629 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5504782 0.82 NLRP3 (0.41) KCNH2NLRP3APPMAP4K4
SCHEMBL4524099 0.79 NLRP3 (0.43) NLRP3APPMAP4K4
SCHEMBL4524773 0.76 NLRP3 (0.46) KCNH2NLRP3APP
SCHEMBL4528798 0.76 RAD52 (0.45) NLRP3APPCYP2D6MAP4K4
Trifluoroacetic Acid SCHEMBL4519544 0.74 APP (0.40) NLRP3APPTLR7
SCHEMBL4519548 0.71 NLRP3 (0.37) NLRP3APPMAP4K4
SCHEMBL13888562 0.71 HRH4 (0.47) KCNH2NLRP3APP
SCHEMBL4517519 0.70 PTPN1 (0.51) KCNH2NLRP3APPMAP4K4
SCHEMBL4526172 0.70 PTPN1 (0.59) NLRP3APPCYP2D6MAP4K4
SCHEMBL4523613 0.67 KCNH2 (0.39) KCNH2NLRP3CYP2D6DRD1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812409-A1 AMINOQUINAZOLINES COMPOUNDS F. Hoffmann-Roche AG (CH) 2007-08-01 EP claimed
WO-2006050843-A1 AMINOQUINAZOLINES COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2006-05-18 WO claimed