SCHEMBL5505243

SCHEMBL5505243

CC(C)Cn1cnc2c(N)nc3ccc(CS(=O)(=O)O)nc3c21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 6/20 0.55
ADORA2A P29274 2/20 0.55
PDE4D Q08499 2/20 0.55
LMNA P02545 1/20 0.55
POLB P06746 1/20 0.55
HRH2 P25021 1/20 0.55
ADRA1D P25100 1/20 0.55
HTR2A P28223 1/20 0.55
ADRA1A P35348 1/20 0.55
NUDT1 P36639 1/20 0.55
HTR2B P41595 1/20 0.55
KCNH2 Q12809 1/20 0.55
MAPK14 Q16539 5/20 0.36
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36
CYP1A2 P05177 1/20 0.34
SLC29A1 Q99808 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5231174 0.89 TLR7 (0.53) TLR7ADORA2APDE4DLMNAPOLB
Epetirimod SCHEMBL4178900 0.80 TLR7 (0.61) TLR7ADORA2APDE4DLMNAPOLB
Epetirimod SCHEMBL4985288 0.80 TLR7 (0.61) TLR7ADORA2APDE4DLMNAPOLB
Epetirimod SCHEMBL4983116 0.79 TLR7 (0.60) TLR7ADORA2APDE4DLMNAPOLB
Epetirimod SCHEMBL4178322 0.79 TLR7 (0.60) TLR7ADORA2APDE4DLMNAPOLB
Imiquimod SCHEMBL9602249 0.76 TLR7 (0.82) TLR7ADORA2APDE4DLMNAPOLB
Epetirimod SCHEMBL29350668 0.75 TLR7 (0.70) TLR7ADORA2APDE4DLMNAPOLB
Epetirimod SCHEMBL544542 0.75 TLR7 (0.70) TLR7ADORA2APDE4DLMNAPOLB
Epetirimod SCHEMBL29454521 0.75 TLR7 (0.70) TLR7ADORA2APDE4DLMNAPOLB
SCHEMBL3862504 0.72 TLR7 (0.73) TLR7ADORA2APDE4DLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833479-A2 1-(2-METHYLPROPYL)-1H-IMIDAZO 4,5-C(1,5 )NAPHTHYRIDIN-4-AMINE ETHANESULFONATE AND 1-(2-METHYLPROPYL)-1H-IMIDAZOÝ4,5-C 1,5 NAPHTHYRIDIN-4-AMINE METHANESULFONATE Takeda Pharmaceutical Company Limited (JP) 2007-09-19 EP disclosed