SCHEMBL5505443

SCHEMBL5505443

NC1=Nc2ccc(Oc3ccccc3)cc2CN1C(CCC(=O)N(CCOCc1ccccc1)C1CCC(OC=O)CC1)C1CCOCC1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 16/20 0.57
REN P00797 1/20 0.56
CTSD P07339 1/20 0.56
KCNH2 Q12809 1/20 0.56
BACE2 Q9Y5Z0 4/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14723920 0.92 BACE1 (0.58) BACE1RENCTSDKCNH2BACE2
SCHEMBL3365249 0.92 BACE1 (0.58) BACE1RENCTSDKCNH2BACE2
SCHEMBL14878030 0.92 BACE1 (0.58) BACE1RENCTSDKCNH2BACE2
SCHEMBL13849173 0.84 BACE1 (0.49) BACE1RENCTSDKCNH2BACE2
SCHEMBL1414460 0.83 BACE1 (0.51) BACE1RENCTSDKCNH2BACE2
SCHEMBL1414274 0.83 BACE1 (0.51) BACE1RENCTSDKCNH2BACE2
SCHEMBL13114565 0.83 BACE1 (0.62) BACE1RENCTSDKCNH2BACE2
SCHEMBL3364771 0.83 BACE1 (0.62) BACE1RENCTSDKCNH2BACE2
SCHEMBL1414117 0.81 BACE1 (0.49) BACE1RENCTSDKCNH2BACE2
SCHEMBL1414119 0.81 BACE1 (0.49) BACE1RENCTSDKCNH2BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1789398-A1 2-AMINO-QUINAZOLINE DERIVATIVES USEFUL AS INHIBITORS OF B-SECRETASE (BACE) JANSSEN PHARMACEUTICA N.V. (BE) 2007-05-30 EP disclosed
WO-2006024932-A1 2-AMINO-QUINAZOLINE DERIVATIVES USEFUL AS INHIBITORS OF B-SECRETASE (BACE) JANSSEN PHARMACEUTICA, N.V. (US) 2006-03-09 WO disclosed