SCHEMBL5506008

SCHEMBL5506008

C[C@H]1CCCN1CCCN1[C]N(CCCN2CCOCC2)CC1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.45
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
KCNH2 Q12809 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP3A4 P08684 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
KEAP1 Q14145 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5507033 0.88 HRH3 (0.42) HRH3
SCHEMBL5502174 0.87 HRH3 (0.44) HRH3
SCHEMBL5508033 0.87 HRH3 (0.42) HRH3
SCHEMBL5508273 0.86 HRH3 (0.37) HRH3CYP2D6
SCHEMBL5506014 0.84 HRH3 (0.47) HRH3CYP1A2CYP2D6KCNH2KEAP1
SCHEMBL5502752 0.84 CXCR4 (0.47) HRH3CHRM2CHRM1
SCHEMBL5506424 0.84 HRH3 (0.41) HRH3
SCHEMBL5505798 0.84 HRH3 (0.41) HRH3
SCHEMBL5506775 0.84 CXCR4 (0.47) HRH3CHRM2CHRM1
SCHEMBL5505523 0.84 HRH3 (0.41) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847530-A1 DIAMINE DERIVATIVE KYOWA HAKKO KOGYO CO., LTD. (JP) 2007-10-24 EP disclosed