Bicarbonate

Bicarbonate

SCHEMBL5506472

C[C@H]1CC[C@H](NC(=N)N)CC1.O=C(O)O

nearest known ligand 0.50

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Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.50
F2 P00734 1/20 0.43
PLG P00747 1/20 0.43
PRSS1 P07477 1/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
ST14 Q9Y5Y6 1/20 0.43
RAB9A P51151 6/20 0.42
NPC1 O15118 4/20 0.42
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ADRA2A P08913 1/20 0.38
MMP2 P08253 1/20 0.38
MMP8 P22894 1/20 0.38
MAPK1 P28482 2/20 0.37
GAA P10253 2/20 0.37
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
TAS1R2 Q8TE23 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL7103163 1.00 EPHX1 (0.50) EPHX1F2PLGPRSS1PRSS2
SCHEMBL19033004 0.92 EPHX1 (0.47) EPHX1F2PLGPRSS1PRSS2
SCHEMBL348519 0.92 EPHX1 (0.47) EPHX1F2PLGPRSS1PRSS2
Hydrochloric Acid SCHEMBL9960143 0.90 EPHX1 (0.45) EPHX1F2PLGPRSS1PRSS2
Hydrochloric Acid SCHEMBL9960141 0.90 EPHX1 (0.45) EPHX1F2PLGPRSS1PRSS2
Acetic Acid SCHEMBL28363861 0.85 POLB (0.39) EPHX1F2PLGPRSS1PRSS2
SCHEMBL1588520 0.80
SCHEMBL20075958 0.80 NOS2 (0.38) EPHX1RAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL3623543 0.79 EPHX1 (0.57) EPHX1F2PLGPRSS1PRSS2
SCHEMBL28310343 0.79 EPHX1 (0.57) EPHX1F2PLGPRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1449828-B1 Guanidinomethyl cyclohexane carboxylic acid ester derivatives NAGASE CHEMTEX CORP (JP) 2007-04-18 EP claimed
EP-0193965-B1 NOVEL GUANIDINOMETHYLCYCLOHEXANCARBOXYLIC ACID COMPOUNDS, PROCESSES FOR PREPARING THEM, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM KANEBO, LTD. (JP) 1988-11-30 EP claimed