SCHEMBL5511565

SCHEMBL5511565

CC(C)C(=O)N(Cc1cccc(Cl)c1Cl)[C@H]1CCN(C(=O)O)C1

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 16/20 0.63
SLC6A2 P23975 15/20 0.63
SLC6A3 Q01959 9/20 0.63
CYP2D6 P10635 4/20 0.63
KCNH2 Q12809 3/20 0.63
CYP3A4 P08684 1/20 0.63
GHSR Q92847 1/20 0.48
UBE2M P61081 2/20 0.43
DCUN1D1 Q96GG9 2/20 0.43
REN P00797 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4485498 0.85 SLC6A2 (0.50) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL5072308 0.84 SLC6A4 (0.76) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL5512041 0.82 SLC6A2 (0.63) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL5506157 0.81 SLC6A2 (0.64) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL4635761 0.78 SLC6A2 (0.62) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL25194484 0.78 GHSR (0.53) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL25265564 0.78 GHSR (0.53) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL5888071 0.72 SLC6A2 (0.45) SLC6A4SLC6A2SLC6A3KCNH2UBE2M
SCHEMBL5511572 0.72 SLC6A2 (0.65) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL4634797 0.72 PDK2 (0.44) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828122-A2 N-PYRROLIDIN-3-YL-AMIDE DERIVATIVES AS SEROTONIN AND NORADRENALIN RE-UPTAKE INHIBITORS Pfizer Limited (GB) 2007-09-05 EP disclosed
WO-2006064351-A2 N-PYRROLIDIN-3-YL-AMIDE DERIVATIVES AS SEROTONIN AND NORADRENALIN RE-UPTAKE INHIBITORS PFIZER LIMITED (GB) 2006-06-22 WO disclosed