SCHEMBL551165

SCHEMBL551165

Clc1ccccc1-c1cccnc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.65
RAB9A P51151 1/20 0.65
TP53 P04637 2/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
NPY5R Q15761 1/20 0.61
CYP2A6 P11509 9/20 0.58
ALDH1A1 P00352 2/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP11B1 P15538 1/20 0.50
MAPK14 Q16539 1/20 0.49
PTGS2 P35354 1/20 0.49
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
ALOX15 P16050 1/20 0.48
HTT P42858 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CNR1 P21554 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30026143 0.84 CYP2A6 (0.70) NPC1RAB9ATP53SMN1; SMN2CYP2A6
SCHEMBL20541087 0.84 CYP2A6 (0.70) NPC1RAB9ATP53SMN1; SMN2CYP2A6
SCHEMBL29412319 0.82 MAPK14 (0.56) NPC1RAB9ATP53SMN1; SMN2NPY5R
SCHEMBL21489665 0.82 NPC1 (0.51) NPC1RAB9ATP53SMN1; SMN2NPY5R
SCHEMBL12853987 0.82 CYP2A6 (0.67) TP53SMN1; SMN2CYP2A6ALDH1A1CYP1A2
SCHEMBL21110859 0.82 CYP2A6 (0.67) TP53SMN1; SMN2CYP2A6ALDH1A1CYP1A2
SCHEMBL27943394 0.82 NPC1 (0.51) NPC1RAB9ATP53SMN1; SMN2NPY5R
SCHEMBL11068804 0.81 NPC1 (0.50) NPC1RAB9ATP53SMN1; SMN2NPY5R
SCHEMBL16110614 0.81 CYP17A1 (0.50) NPC1RAB9ATP53SMN1; SMN2NPY5R
SCHEMBL16513266 0.81 NPY5R (0.67) NPC1RAB9ATP53SMN1; SMN2NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210221784-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PAIN UNIVERSITÉ DE STRASBOURG (FR) 2021-07-22 US disclosed
WO-2019022435-A1 COMPOUND FOR ORGANIC ELECTRONIC DEVICE, ORGANIC ELECTRONIC DEVICE USING SAME, AND ELECTRONIC APPARATUS THEREOF 덕산네오룩스 주식회사 2019-01-31 WO disclosed
CN-108997342-A A kind of two fluorene compound of more azaspiros and the organic electro-optic device containing the compound 上海大学 2018-12-14 CN disclosed
EP-1572681-B1 3-SUBSTITUTED-4-PYRIMIDONE DERIVATIVES MITSUBISHI TANABE PHARMA CORP (JP) 2014-01-22 EP disclosed
US-8110642-B2 Synthesis of vinylphenylpyridine and living anionic polymerization GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2012-02-07 US disclosed
CN-1726209-B 3-substituted-4-pyrimidone derivatives SANOFI AVENTIS 2011-04-13 CN disclosed
US-7683069-B2 3-substituted-4-pyrimidone derivatives MITSUBISHI TANABE PHARMA CORPORATION (JP) 2010-03-23 US disclosed
US-20090105416-A1 Synthesis of Vinylphenylpyridine and Living Anionic Polymerization GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-23 US disclosed
WO-2007129810-A1 SYNTHESIS OF VINYLPHENYLPYRIDINE AND LIVING ANIONIC POLYMERIZATION GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2007-11-15 WO disclosed
US-20070142409-A1 3-Substituted-4-pyrimidone derivatives MITSUBISHI PHARMA CORPORATION OF OSAKA JAPAN 2007-06-21 US disclosed
CN-1726209-A 3-substituted-4-pyrimidone derivatives SANOFI AVENTIS (JP) 2006-01-25 CN disclosed
EP-1572681-A1 3-SUBSTITUTED-4-PYRIMIDONE DERIVATIVES MITSUBISHI PHARMA CORPORATION (JP) 2005-09-14 EP disclosed
WO-2004055007-A1 3-SUBSTITUTED-4-PYRIMIDONE DERIVATIVES MITSUBISHI PHARMA CORPORATION (JP) 2004-07-01 WO disclosed
EP-1381606-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 2004-01-21 EP disclosed
WO-2002074773-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 2002-09-26 WO disclosed
US-4244953-A Substituted 6-phenyl-5,6,7,8-tetrahydro-1,2,4-triazolo-[4,3-a]pyridines AMERICAN CYANAMID COMPANY (US) 1981-01-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210221784-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PAIN ACHE, TRPV1, OPRL1 NPC1 2638/4885RAB9A 3565/4885TP53 4089/4885
US-20090105416-A1 Synthesis of Vinylphenylpyridine and Living Anionic Polymerization PBRM1, MVD, PCBP1 NPC1 4810/4885RAB9A 4209/4885TP53 2979/4885
US-20070142409-A1 3-Substituted-4-pyrimidone derivatives TTBK1, MAPT, TTBK2 NPC1 2202/4885RAB9A 3514/4885TP53 748/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.