SCHEMBL5514820

SCHEMBL5514820

CCCCCCCC/C=C\CCCCCCCCOC(CC)(OCCCCCCCC/C=C\CCCCCCCC)[N+](C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LPAR3 Q9UBY5 4/20 0.44
LPAR2 Q9HBW0 3/20 0.44
LPAR1 Q92633 2/20 0.44
FAAH O00519 2/20 0.41
TRPV1 Q8NER1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8715666 0.98 LPAR3 (0.42) LPAR3LPAR2LPAR1FAAHTRPV1
SCHEMBL18837389 0.85 LPAR3 (0.42) LPAR3LPAR2LPAR1FAAHTRPV1
SCHEMBL1906179 0.76 LPAR2 (0.44) LPAR3LPAR2LPAR1FAAHTRPV1
SCHEMBL6831358 0.76 LPAR2 (0.44) LPAR3LPAR2LPAR1FAAHTRPV1
SCHEMBL1933828 0.76 LPAR3 (0.44) LPAR3LPAR2LPAR1FAAHTRPV1
SCHEMBL18184028 0.76 LPAR2 (0.50) LPAR3LPAR2LPAR1FAAHTRPV1
SCHEMBL16311960 0.76 LPAR2 (0.50) LPAR3LPAR2LPAR1FAAHTRPV1
SCHEMBL27094088 0.75 LPAR3 (0.46) LPAR3LPAR2LPAR1FAAHTRPV1
SCHEMBL20500071 0.74 LPAR3 (0.49) LPAR3LPAR2LPAR1FAAHTRPV1
SCHEMBL20500069 0.74 LPAR3 (0.49) LPAR3LPAR2LPAR1FAAHTRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946153-A1 HOMOGENEOUSLY CHARGED PARTICULATE VECTOR AND PHARMACEUTICAL OR COSMETIC COMPOSITION CONTAINING SAME BIOVECTOR THERAPEUTICS SA (FR) 1999-10-06 EP claimed
WO-1998029102-A1 HOMOGENEOUSLY CHARGED PARTICULATE VECTOR AND PHARMACEUTICAL OR COSMETIC COMPOSITION CONTAINING SAME BIOVECTOR THERAPEUTICS S.A. (FR) 1998-07-09 WO claimed
US-9238056-B2 Cyclic peptide and conjugate thereof for binding to keratinocytes LEO PHARMA A/S (DK) 2016-01-19 US disclosed
US-20140023700-A1 CYCLIC PEPTIDE AND CONJUGATE THEREOF FOR BINDING TO KERATINOCYTES LEO PHARMA A/S (DK) 2014-01-23 US disclosed
EP-2678350-A1 A CYCLIC PEPTIDE AND CONJUGATE THEREOF FOR BINDING TO KERATINOCYTES Leo Pharma A/S (DK) 2014-01-01 EP disclosed
WO-2012113803-A1 A CYCLIC PEPTIDE AND CONJUGATE THEREOF FOR BINDING TO KERATINOCYTES LEO PHARMA A/S (DK) 2012-08-30 WO disclosed
US-20070116767-A1 Chitosan-microparticles for ifn gene delivery UNIVERSITY OF SOUTH FLORIDA 2007-05-24 US disclosed
WO-2005105136-A9 NANOGENE THERAPY FOR CELL PROLIFERATION DISORDERS UNIV SOUTH FLORIDA (US) 2006-03-02 WO disclosed
US-20050266093-A1 Nanogene therapy for cell proliferation disorders UNIVERSITY OF SOUTH FLORIDA 2005-12-01 US disclosed
EP-1594547-A2 CHITOSAN-MICROPARTICLES FOR IFN GENE DELIVERY University Of South Florida Research Foundation, Inc. (US) 2005-11-16 EP disclosed
WO-2005105136-A1 NANOGENE THERAPY FOR CELL PROLIFERATION DISORDERS UNIVERSITY OF SOUTH FLORIDA (US) 2005-11-10 WO disclosed
WO-2004074314-A2 CHISTOSAN-MICROPARTICLES FOR IFN GENE DELIVERY UNIVERSITY OF SOUTH FLORIDA (US) 2004-09-02 WO disclosed
EP-0946153-A1 HOMOGENEOUSLY CHARGED PARTICULATE VECTOR AND PHARMACEUTICAL OR COSMETIC COMPOSITION CONTAINING SAME BIOVECTOR THERAPEUTICS SA (FR) 1999-10-06 EP disclosed
WO-1998029102-A1 HOMOGENEOUSLY CHARGED PARTICULATE VECTOR AND PHARMACEUTICAL OR COSMETIC COMPOSITION CONTAINING SAME BIOVECTOR THERAPEUTICS S.A. (FR) 1998-07-09 WO disclosed