SCHEMBL5516875

SCHEMBL5516875

Cc1ccc(-c2ccc3nccc(Nc4ccc(N5CCC(N(S(C)(=O)=O)S(C)(=O)=O)C5)cc4)c3c2)cc1F

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 17/20 0.51
MELK Q14680 1/20 0.42
TGFBR1 P36897 1/20 0.40
RAF1 P04049 1/20 0.39
BRAF P15056 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4146627 0.90 MAPKAPK2 (0.56) MAPKAPK2MELK
SCHEMBL5506286 0.86 MAPKAPK2 (0.53) MAPKAPK2
SCHEMBL5506279 0.86 MAPKAPK2 (0.53) MAPKAPK2
SCHEMBL4140347 0.84 MAPKAPK2 (0.55) MAPKAPK2MELK
SCHEMBL4154685 0.83 MAPKAPK2 (0.56) MAPKAPK2
SCHEMBL4154112 0.81 MAPKAPK2 (0.56) MAPKAPK2MELK
SCHEMBL4145451 0.81 MAPKAPK2 (0.55) MAPKAPK2MELK
SCHEMBL4143228 0.80 MAPKAPK2 (0.68) MAPKAPK2
SCHEMBL4141129 0.79 MAPKAPK2 (0.54) MAPKAPK2MELKRAF1BRAF
SCHEMBL4161518 0.79 MAPKAPK2 (0.55) MAPKAPK2MELK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781293-A1 QUINOLINE- AND ISOQUINOLINE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF Amphora Discovery Corporation (US) 2007-05-09 EP disclosed
WO-2005120509-A1 QUINOLINE- AND ISOQUINOLINE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-12-22 WO disclosed