SCHEMBL5520004

SCHEMBL5520004

CC(C)C(C(=O)O)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.66
BACE1 P56817 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP1A2 P05177 1/20 0.50
GAA P10253 1/20 0.50
CYP2C9 P11712 1/20 0.50
PKM P14618 1/20 0.50
CYP2C19 P33261 1/20 0.50
AKR1C3 P42330 1/20 0.49
AKR1C2 P52895 1/20 0.49
MMP2 P08253 2/20 0.46
MMP3 P08254 2/20 0.46
MMP13 P45452 2/20 0.46
ADAMTS4 O75173 1/20 0.46
MMP1 P03956 1/20 0.46
MMP7 P09237 1/20 0.46
MMP9 P14780 1/20 0.46
PDCD1 Q15116 1/20 0.46
CD274 Q9NZQ7 1/20 0.46
ACP3 P15309 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5158960 0.87 CYP2D6 (0.73) PTGS2CYP2D6AKR1C3AKR1C2
SCHEMBL66944 0.87 CYP2D6 (0.73) PTGS2CYP2D6AKR1C3AKR1C2
SCHEMBL193565 0.87 CYP2D6 (0.73) PTGS2CYP2D6AKR1C3AKR1C2
SCHEMBL29279091 0.86 PTGS2 (0.63) PTGS2BACE1CYP2D6CYP1A2GAA
Hydrochloric Acid SCHEMBL10582883 0.85 CYP2D6 (0.70) PTGS2CYP2D6AKR1C3AKR1C2
Hydrochloric Acid SCHEMBL10872012 0.85 CYP2D6 (0.70) PTGS2CYP2D6AKR1C3AKR1C2
SCHEMBL289164 0.85 PTGS2 (0.61) PTGS2BACE1CYP2D6CYP1A2GAA
SCHEMBL5515246 0.82 KMT2A (0.65) PTGS2BACE1CYP1A2GAACYP2C9
SCHEMBL24894125 0.80 PTGS2 (0.56) PTGS2BACE1CYP2D6CYP1A2GAA
SCHEMBL24894120 0.80 PTGS2 (0.56) PTGS2BACE1CYP2D6CYP1A2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed