SCHEMBL5521147

SCHEMBL5521147

COC(=O)[C@@H](Cc1ccccc1)NC(=O)c1cc(C)c(C)n(CC2CCCCC2)c1=O

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 8/20 0.60
CNR1 P21554 7/20 0.60
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
PKM P14618 1/20 0.47
ATM Q13315 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
GAA P10253 2/20 0.46
TACR3 P29371 1/20 0.45
NLRP3 Q96P20 2/20 0.43
ACE P12821 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2747934 1.00 CNR2 (0.60) CNR2CNR1KDM4EALDH1A1PKM
SCHEMBL2745651 0.92 CNR1 (0.53) CNR2CNR1NLRP3
SCHEMBL5517849 0.92 CNR1 (0.71) CNR2CNR1ALDH1A1L3MBTL1GAA
SCHEMBL5524504 0.92 CNR1 (0.71) CNR2CNR1ALDH1A1L3MBTL1GAA
SCHEMBL14472292 0.87 CNR2 (0.57) CNR2CNR1KDM4EALDH1A1PKM
SCHEMBL2746851 0.87 CNR1 (0.46) CNR2CNR1KDM4EALDH1A1PKM
SCHEMBL14679033 0.85 CNR2 (0.84) CNR2CNR1
SCHEMBL2746665 0.85 CNR2 (0.84) CNR2CNR1
SCHEMBL2746797 0.85 TAS1R3 (0.47) CNR2CNR1
SCHEMBL5524996 0.85 CNR2 (0.44) CNR2CNR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed