SCHEMBL5530322

SCHEMBL5530322

CON(C(=O)C1CCCC(CNC(=O)OC(C)(C)C)C1)c1ccnc2cccnc12

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACACB O00763 11/20 0.40
ACACA Q13085 8/20 0.40
KDM4E B2RXH2 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CKS1B P61024 1/20 0.35
SKP1 P63208 1/20 0.35
SKP2 Q13309 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
PBK Q96KB5 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
DRD2 P14416 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5432646 0.89 CNR1 (0.40) ACACBACACAKDM4ECKS1BSKP1
SCHEMBL5636825 0.80 JAK1 (0.40) CKS1BSKP1SKP2DRD2
SCHEMBL5636179 0.80 KDM4D (0.33) KDM4ETDP1
SCHEMBL5260297 0.80 KDM4D (0.33) KDM4ETDP1
SCHEMBL3577407 0.79 KDM4D (0.32) KDM4ETDP1
SCHEMBL5506645 0.76 KDM4E (0.41) ACACBACACAKDM4ECKS1BSKP1
SCHEMBL633008 0.75 USP30 (0.42) KDM4EADORA2AADORA2B
SCHEMBL5530317 0.72 KCNH2 (0.47) ACACBACACACKS1BSKP1SKP2
SCHEMBL5261192 0.71 KDM4E (0.33) KDM4ETDP1
SCHEMBL2369250 0.70 ACACB (0.48) ACACBACACACKS1BSKP1SKP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799676-A2 NEW BICYCLIC ANTIBIOTICS Actelion Pharmaceuticals Ltd. (CH) 2007-06-27 EP disclosed
WO-2006032466-A2 NEW BICYCLIC ANTIBIOTICS ACTELION PHARMACEUTICALS LTD (CH) 2006-03-30 WO disclosed