SCHEMBL5540840

SCHEMBL5540840

O=C(NCCCN1CCCC1=O)c1ccccc1C(=O)NCCn1c(=O)c(C(=O)NCCCN2CCCC2=O)c(O)c2ncc(Cc3ccc(F)cc3)cc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
KDM4E B2RXH2 3/20 0.49
GAA P10253 2/20 0.49
HPGD P15428 2/20 0.49
HSD17B10 Q99714 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.47
RXFP1 Q9HBX9 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
CYP2C19 P33261 1/20 0.43
TYRO3 Q06418 3/20 0.42
TSHR P16473 1/20 0.42
LMNA P02545 1/20 0.42
CASK O14936 1/20 0.42
MERTK Q12866 1/20 0.42
GPR52 Q9Y2T5 1/20 0.41
FSHR P23945 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
MAPK1 P28482 1/20 0.41
CREBBP Q92793 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5539930 0.93 CYP2C19 (0.46) ALDH1A1KDM4EGAAHPGDHSD17B10
SCHEMBL5547092 0.93 CYP2C19 (0.46) ALDH1A1KDM4EGAAHPGDHSD17B10
SCHEMBL5543248 0.93 CYP2C19 (0.45) ALDH1A1KDM4EGAAHPGDHSD17B10
SCHEMBL5546009 0.93 CYP2C19 (0.46) ALDH1A1KDM4EGAAHPGDHSD17B10
SCHEMBL5547250 0.92 CYP2C19 (0.44) ALDH1A1KDM4EGAAHPGDHSD17B10
SCHEMBL5539125 0.92 CYP2C19 (0.45) ALDH1A1KDM4EGAAHPGDHSD17B10
SCHEMBL5541025 0.91 CYP2C19 (0.45) ALDH1A1KDM4EGAAHPGDHSD17B10
SCHEMBL16009342 0.91 ALDH1A1 (0.42) ALDH1A1KDM4EGAAHPGDHSD17B10
SCHEMBL5538498 0.91 CYP2C19 (0.44) ALDH1A1KDM4EGAAHPGDHSD17B10
SCHEMBL5538937 0.90 RXFP1 (0.42) ALDH1A1KDM4EGAAHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070124152-A1 Hiv Integrase Inhibitors GLAXOSMITHKLINE LLC 2007-05-31 US disclosed