SCHEMBL5547149

SCHEMBL5547149

[CH2]CCC(c1cccnc1)n1ccnn1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 0.44
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
CFTR P13569 1/20 0.37
GOPC Q9HD26 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.35
KDM4E B2RXH2 2/20 0.34
TBXAS1 P24557 1/20 0.33
CHRNA7 P36544 1/20 0.33
GRM8 O00222 1/20 0.32
GRM4 Q14833 1/20 0.32
KCNA5 P22460 2/20 0.32
LMNA P02545 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KCNH2 Q12809 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27684288 0.82 CYP19A1 (0.46) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL5550616 0.75 CYP17A1 (0.47) CYP19A1KCNH2ALDH1A1
SCHEMBL1243818 0.73 CYP19A1 (0.49) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL29273163 0.70 CYP19A1 (0.57) CYP19A1
SCHEMBL28028213 0.68 CFTR (0.46) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL1240484 0.68 KCNA5 (0.54) CYP19A1SMN1; SMN2KCNA5KCNH2
SCHEMBL27475767 0.68 HRH1 (0.40) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL9965186 0.68 CYP19A1 (0.43) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL20773275 0.67 CYP19A1 (0.62) CYP19A1
SCHEMBL401391 0.67 CYP19A1 (0.53) CYP19A1SLC6A2SLC6A4SLC6A3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1830858-A2 3, 6-BICYCLOLIDES Enanta Pharmaceuticals, Inc. (US) 2007-09-12 EP disclosed
WO-2006063039-A2 3, 6-BICYCLOLIDES ENANTA PHARMACEUTICALS, INC. (US) 2006-06-15 WO disclosed