SCHEMBL9965186

SCHEMBL9965186

Nc1ccc(C(C(c2cccnc2)c2cccnc2)n2ccnn2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 6/20 0.43
CFTR P13569 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
GOPC Q9HD26 1/20 0.36
CYP17A1 P05093 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
KDM4E B2RXH2 1/20 0.33
NOTUM Q6P988 1/20 0.32
KCNN4 O15554 1/20 0.31
KCNA5 P22460 1/20 0.31
CYP3A4 P08684 1/20 0.30
CYP3A5 P20815 1/20 0.30
MEN1 O00255 1/20 0.30
PSIP1 O75475 1/20 0.30
AXL P30530 1/20 0.30
MKNK1 Q9BUB5 1/20 0.30
MKNK2 Q9HBH9 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1243818 0.90 CYP19A1 (0.49) CYP19A1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL9965131 0.86 CYP19A1 (0.41) CYP19A1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL1242629 0.84 CYP19A1 (0.57) CYP19A1CYP17A1KCNA5CYP3A4
SCHEMBL1243320 0.78 CYP19A1 (0.44) CYP19A1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL1242145 0.77 CYP19A1 (0.45) CYP19A1CYP17A1KCNA5ALDH1A1
SCHEMBL9965132 0.76 KCNA5 (0.40) CYP19A1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL1242375 0.72 CFTR (0.41) CYP19A1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL4047293 0.71 CFTR (0.43) CYP19A1CFTRSLC6A2SLC6A4SLC6A3
SCHEMBL9965135 0.70 CYP19A1 (0.70) CYP19A1SMN1; SMN2NOTUMMEN1ALDH1A1
SCHEMBL27684288 0.70 CYP19A1 (0.46) CYP19A1CFTRSLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082746-A2 METALLOENZYME INHIBITOR COMPOUNDS VIAMET PHARMACEUTICALS, INC. (US) 2012-06-21 WO disclosed