SCHEMBL5547151

SCHEMBL5547151

Cc1cccc(-c2cc(CCCO)nc(C#N)n2)c1C

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSK P43235 20/20 0.55
KCNH2 Q12809 4/20 0.55
CTSS P25774 15/20 0.46
CTSL P07711 2/20 0.41
CTSB P07858 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4447789 0.86 CTSK (0.62) CTSKCTSS
SCHEMBL4442745 0.77 CTSK (0.74) CTSKKCNH2CTSSCTSLCTSB
SCHEMBL5022259 0.77 CTSK (0.48) CTSKKCNH2CTSSCTSLCTSB
SCHEMBL13707273 0.76 CTSK (0.69) CTSKKCNH2CTSSCTSLCTSB
SCHEMBL4451832 0.73 CTSK (0.79) CTSKKCNH2CTSSCTSLCTSB
SCHEMBL4444381 0.71 CTSK (1.00) CTSKKCNH2CTSSCTSLCTSB
SCHEMBL13709386 0.70 CTSK (0.52) CTSKKCNH2CTSSCTSLCTSB
SCHEMBL5017270 0.67 CTSK (0.42) CTSKKCNH2CTSSCTSLCTSB
SCHEMBL5798709 0.66 CTSK (0.71) CTSKKCNH2CTSSCTSB
SCHEMBL4442123 0.65 TLR8 (0.34) CTSKKCNH2CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758870-A1 4-PHENYL-PYRIMIDINE-2-CARBONITRILE DERIVATIVES N.V. Organon (NL) 2007-03-07 EP disclosed
WO-2005121106-A1 4-PHENYL-PYRIMIDINE-2-CARBONITRILE DERIVATIVES N.V. ORGANON (NL) 2005-12-22 WO disclosed