SCHEMBL5547995

SCHEMBL5547995

COc1ccc(C(=O)N2C=C3CN=C(NC(=O)c4cccc(Cl)c4)N=C3CC2)cc1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
POLB P06746 2/20 0.41
MEN1 O00255 2/20 0.41
ALDH1A1 P00352 3/20 0.41
ATM Q13315 1/20 0.40
PDE4D Q08499 2/20 0.40
PTGS2 P35354 1/20 0.40
USP2 O75604 2/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39
GRM5 P41594 1/20 0.39
PDE4B Q07343 1/20 0.39
MAPK14 Q16539 1/20 0.39
KDM4E B2RXH2 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
ROCK2 O75116 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5537982 0.78 NPC1 (0.42) KMT2APOLBMEN1ALDH1A1RAB9A
SCHEMBL5547993 0.74 GRM5 (0.41) ALDH1A1PDE4DUSP2MAPK1GRM5
SCHEMBL5548545 0.71 SIRT2 (0.42) KMT2APOLBMEN1ATMTP53
SCHEMBL5538068 0.71 MAPT (0.39) KMT2ARAB9AKDM4EMAPT
SCHEMBL5546587 0.68 ALDH1A1 (0.45) KMT2AMEN1ALDH1A1USP2MAPK1
SCHEMBL3531464 0.67 PDGFRB (0.61) POLBMAPK1PDE4BKDM4EMAPT
SCHEMBL14553659 0.67 MAOB (0.64) KMT2AALDH1A1PDE4DPTGS2PDE4B
SCHEMBL5546575 0.66 ADORA2A (0.36) KMT2APOLBMEN1MAPT
SCHEMBL5546854 0.66 CYP2C19 (0.40) KMT2AMEN1ALDH1A1MAPK1RAB9A
SCHEMBL5546893 0.64 MAPT (0.40) KMT2AMEN1ALDH1A1USP2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed