SCHEMBL5548893

SCHEMBL5548893

CC(C)(C)c1cn2c(=O)[nH]nc2c(NCCOc2ccccc2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 5/20 0.49
GSK3B P49841 5/20 0.49
GPR84 Q9NQS5 2/20 0.41
KMT2A Q03164 2/20 0.39
ADORA1 P30542 2/20 0.39
ATM Q13315 1/20 0.38
MPO P05164 1/20 0.38
AURKA O14965 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
RAB9A P51151 2/20 0.36
LMNA P02545 2/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPC1 O15118 1/20 0.36
POLB P06746 1/20 0.36
CASP3 P42574 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3527708 0.92 GSK3A (0.57) GSK3AGSK3BKMT2ARAB9ALMNA
SCHEMBL3529920 0.91 GSK3A (0.61) GSK3AGSK3BKMT2ARAB9ALMNA
SCHEMBL3525341 0.91 GSK3B (0.48) GSK3AGSK3BAURKACYP2D6RAB9A
SCHEMBL5549831 0.90 GSK3A (0.50) GSK3AGSK3BRAB9ALMNAHTT
SCHEMBL3521643 0.89 GSK3A (0.43) GSK3AGSK3BKMT2AAURKACYP2D6
SCHEMBL3530232 0.89 GSK3A (0.46) GSK3AGSK3BGPR84AURKACYP3A4
SCHEMBL5549009 0.87 GSK3A (0.43) GSK3AGSK3BKMT2AADORA1CYP3A4
SCHEMBL5550212 0.87 GSK3A (0.44) GSK3AGSK3BKMT2ALMNAHTT
SCHEMBL5548604 0.86 GSK3A (0.48) GSK3AGSK3BAURKACYP3A4CYP2D6
SCHEMBL5548595 0.85 GSK3B (0.48) GSK3AGSK3BLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed