SCHEMBL5548604

SCHEMBL5548604

Cc1ccc(OCCNc2nc(C(C)(C)C)cn3c(=O)[nH]nc23)cn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 15/20 0.48
GSK3B P49841 15/20 0.48
AURKA O14965 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
RAB29 O14966 1/20 0.41
FYN P06241 1/20 0.41
YES1 P07947 1/20 0.41
LYN P07948 1/20 0.41
FGFR1 P11362 1/20 0.41
SRC P12931 1/20 0.41
KDR P35968 1/20 0.41
AURKB Q96GD4 1/20 0.41
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3527708 0.90 GSK3A (0.57) GSK3AGSK3BLMNAHTTRAB9A
SCHEMBL3521643 0.88 GSK3A (0.43) GSK3AGSK3BAURKACYP1A2SMN1; SMN2
SCHEMBL3529920 0.87 GSK3A (0.61) GSK3AGSK3BLMNAHTTRAB9A
SCHEMBL5549831 0.86 GSK3A (0.50) GSK3AGSK3BLMNAHTTRAB9A
SCHEMBL5550070 0.86 GSK3A (0.50) GSK3AGSK3BLMNAHTTRAB9A
SCHEMBL5548893 0.86 GSK3A (0.49) GSK3AGSK3BAURKACYP3A4LMNA
SCHEMBL3525341 0.85 GSK3B (0.48) GSK3AGSK3BAURKALMNAHTT
SCHEMBL3526786 0.84 GSK3B (0.56) GSK3AGSK3B
SCHEMBL5548595 0.84 GSK3B (0.48) GSK3AGSK3BLMNASMN1; SMN2
SCHEMBL5545002 0.83 GSK3A (0.51) GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed