SCHEMBL5550007

SCHEMBL5550007

CC(C)(C)c1cn2c(=O)[nH]nc2c(NCCN2CCCC2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT2B Q92831 4/20 0.39
IKBKB O14920 1/20 0.37
CHUK O15111 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KMT5A Q9NQR1 1/20 0.35
MAPT P10636 2/20 0.35
APAF1 O14727 1/20 0.35
NPC1 O15118 1/20 0.35
NSD2 O96028 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
BLM P54132 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
ILK Q13418 1/20 0.35
TOP2A P11388 1/20 0.34
RAD52 P43351 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5548887 0.99 KAT2B (0.40) KAT2BIKBKBCHUKMEN1KMT2A
SCHEMBL5549838 0.93 PGK1 (0.40) KAT2BKMT5ATLR7GSK3AGSK3B
SCHEMBL5549410 0.90 TLR9 (0.43) MEN1KMT2AAPAF1NSD2HTT
SCHEMBL5549394 0.87 PGK1 (0.39) KAT2BKMT5ATLR9TLR7GSK3A
SCHEMBL3526664 0.84 GAA (0.45) MEN1KMT2AMAPTNPC1RAB9A
SCHEMBL5545590 0.82 GSK3B (0.35) GSK3AGSK3B
SCHEMBL3521775 0.82 GSK3B (0.36) IKBKBCHUKGSK3AGSK3B
SCHEMBL3529268 0.82 ADORA1 (0.37) GSK3AGSK3B
SCHEMBL5548632 0.81 KDM1A (0.40) KAT2BMEN1KMT2ANPC1RAB9A
SCHEMBL5543598 0.81 HSD17B10 (0.43) KAT2BGSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed