SCHEMBL5551100

SCHEMBL5551100

O=C=Nc1ccccc1/C=C/c1ccccc1N=C=O

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.50
NFE2L2 Q16236 3/20 0.36
TRPA1 O75762 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
THRB P10828 1/20 0.35
BLM P54132 1/20 0.35
KMT2A Q03164 1/20 0.35
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
CA12 O43570 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3099538 1.00 CYP3A4 (0.50) CYP3A4NFE2L2TRPA1TDP1MEN1
SCHEMBL31168163 1.00 CYP3A4 (0.50) CYP3A4NFE2L2TRPA1TDP1MEN1
SCHEMBL11022955 0.90 NFE2L2 (0.46) CYP3A4NFE2L2TRPA1MEN1LMNA
SCHEMBL11022950 0.90 NFE2L2 (0.46) CYP3A4NFE2L2TRPA1MEN1LMNA
SCHEMBL29127235 0.89 CYP3A4 (0.50) CYP3A4TRPA1MEN1LMNABLM
SCHEMBL29127250 0.89 APOBEC3A (0.42) CYP3A4NFE2L2TRPA1MEN1LMNA
SCHEMBL5402133 0.88 CYP3A4 (0.48) CYP3A4TRPA1TDP1MEN1LMNA
SCHEMBL5402136 0.88 CYP3A4 (0.48) CYP3A4TRPA1TDP1MEN1LMNA
SCHEMBL10890112 0.86 CYP3A4 (0.50) CYP3A4TRPA1TDP1MEN1LMNA
SCHEMBL11683007 0.86 CYP3A4 (0.39) CYP3A4NFE2L2TRPA1TDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817615-A1 SUN PROTECTION FILM WHICH ABSORBS INFRARED RADIATION Air Products and Chemicals, Inc. (US) 2007-08-15 EP disclosed
WO-2006058870-A1 SUN PROTECTION FILM WHICH ABSORBS INFRARED RADIATION AIR PRODUCTS AND CHEMICALS, INC. (US) 2006-06-08 WO disclosed
EP-0910597-A1 PROCESS FOR PREPARING CELLULAR POLYURETHANE ELASTOMERS BASED ON 3,3'-DIMETHOXY-4,4'DIISOCYANATO-DIPHENYL AND/OR 4,4'-STILBENE-DIISOCYANATE BASF AKTIENGESELLSCHAFT (DE) 1999-04-28 EP disclosed
WO-1998002477-A1 PROCESS FOR PREPARING CELLULAR POLYURETHANE ELASTOMERS BASED ON 3,3'-DIMETHOXY-4,4'DIISOCYANATO-DIPHENYL AND/OR 4,4'-STILBENE-DIISOCYANATE BASF AKTIENGESELLSCHAFT (DE) 1998-01-22 WO disclosed
EP-0011784-B1 SUSPENSIONS OF AROMATIC ISOCYANATOSULFONIC-ACID URETDIONES IN ORGANIC POLYISOCYANATES AND PROCESS FOR THEIR PREPARATION BAYER AG (DE) 1982-03-24 EP disclosed
EP-0000723-B1 POLYHYDROXY COMPOUNDS CONTAINING URETHANE-ARYL-SULFONIC ACID-HYDROXYALKYL ESTER GROUPS, PROCESS FOR THEIR PREPARATION AND THEIR USE AS REACTION COMPONENTS FOR THE PREPARATION OF POLYURETHANE RESINS BAYER AG (DE) 1981-01-07 EP disclosed
EP-0004277-B1 PROCESS TO IMPROVE THE STORAGE STABILITY OF FINELY DISPERSED AROMATIC ISOCYANATOSULFONIC ACIDS AND THE CORRESPONDING STABILIZED PREPARATIONS BAYER AG (DE) 1980-12-10 EP disclosed