SCHEMBL5551950

SCHEMBL5551950

CCCc1ccc(NC(=O)CC(C)=O)cc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.81
MAPT P10636 1/20 0.57
TSHR P16473 1/20 0.57
HDAC3 O15379 1/20 0.55
HDAC4 P56524 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC7 Q8WUI4 1/20 0.55
HDAC2 Q92769 1/20 0.55
HDAC10 Q969S8 1/20 0.55
HDAC11 Q96DB2 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
HDAC9 Q9UKV0 1/20 0.55
HDAC5 Q9UQL6 1/20 0.55
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA4 P22748 1/20 0.54
CA7 P43166 1/20 0.54
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9312694 0.91 POLB (0.67) POLBHDAC3HDAC4HDAC1HDAC7
SCHEMBL9429642 0.90 POLB (1.00) POLBMAPTTSHRHDAC3HDAC4
SCHEMBL7057797 0.88 POLB (0.91) POLBCA1CA2NPC1RAB9A
SCHEMBL13239485 0.87 POLB (0.88) POLBCA1CA2NPC1RAB9A
SCHEMBL7056819 0.87 POLB (0.88) POLBCA1CA2NPC1RAB9A
SCHEMBL11983728 0.86 POLB (0.71) POLBMAPTTSHRHDAC3HDAC4
SCHEMBL17874906 0.86 POLB (0.61) POLBHDAC3HDAC4HDAC1HDAC7
SCHEMBL10117151 0.85 POLB (0.60) POLBMAPTHDAC3HDAC4HDAC1
SCHEMBL7055067 0.85 POLB (0.70) POLBMAPTTSHRHDAC3HDAC4
SCHEMBL593172 0.84 MAPT (0.74) POLBMAPTTSHRCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1742924-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-01-17 EP disclosed
WO-2005108376-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2005-11-17 WO disclosed