SCHEMBL5552182

SCHEMBL5552182

NC1CCC(c2cccc(F)c2F)CN(C(=O)OCc2ccccc2)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.46
CYP2C19 P33261 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
JAK2 O60674 2/20 0.41
JAK1 P23458 2/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CNR2 P34972 1/20 0.40
KDM1A O60341 2/20 0.39
MAOA P21397 2/20 0.39
MAOB P27338 2/20 0.39
TMEM97 Q5BJF2 2/20 0.39
SIGMAR1 Q99720 2/20 0.39
DPP4 P27487 1/20 0.39
PDE4B Q07343 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2C P18825 1/20 0.39
HRH2 P25021 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1434918 1.00 SMN1; SMN2 (0.46) SMN1; SMN2CYP2C19NPC1RAB9AJAK2
SCHEMBL4564213 0.80 BCL9 (0.52) SMN1; SMN2CYP2C19NPC1RAB9AJAK2
SCHEMBL1435091 0.80 PDE4B (0.47) KMT2ADPP4PDE4BUSP30
SCHEMBL19404905 0.79 SMN1; SMN2 (0.57) SMN1; SMN2CYP2C19NPC1RAB9AJAK2
SCHEMBL16653836 0.78 SMN1; SMN2 (0.58) SMN1; SMN2CYP2C19NPC1RAB9AJAK2
SCHEMBL14428334 0.78 SMN1; SMN2 (0.58) SMN1; SMN2CYP2C19NPC1RAB9AJAK2
SCHEMBL15379354 0.78 SMN1; SMN2 (0.61) SMN1; SMN2CYP2C19NPC1RAB9AMEN1
SCHEMBL654999 0.76 SMN1; SMN2 (0.60) SMN1; SMN2CYP2C19NPC1RAB9AJAK2
SCHEMBL764193 0.76 SMN1; SMN2 (0.60) SMN1; SMN2CYP2C19NPC1RAB9AJAK2
SCHEMBL12791106 0.76 SMN1; SMN2 (0.60) SMN1; SMN2CYP2C19NPC1RAB9AJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1804919-A2 CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2007-07-11 EP disclosed
WO-2006047196-A2 CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2006-05-04 WO disclosed