SCHEMBL5554293

SCHEMBL5554293

CCCCNC(=O)Cc1c(C)n(C(=S)c2ccc(CC)cc2)c2cc(Cl)c(O)cc12

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.50
CA2 P00918 3/20 0.50
PTGS2 P35354 14/20 0.48
PTGS1 P23219 6/20 0.47
HRH4 Q9H3N8 1/20 0.43
HDAC3 O15379 3/20 0.41
HDAC1 Q13547 3/20 0.41
HDAC8 Q9BY41 3/20 0.41
HDAC6 Q9UBN7 3/20 0.41
HDAC2 Q92769 1/20 0.41
CA12 O43570 2/20 0.41
CA4 P22748 2/20 0.41
CA9 Q16790 2/20 0.41
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6424039 0.94 PTGS2 (0.49) CA1CA2PTGS2PTGS1HRH4
SCHEMBL5553909 0.88 PTGS2 (0.45) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL5560111 0.84 PTGS2 (0.66) CA1CA2PTGS2PTGS1HRH4
SCHEMBL5554102 0.84 PTGS2 (0.59) CA1CA2PTGS2PTGS1HRH4
SCHEMBL5560561 0.84 PTGS2 (0.51) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL5560837 0.84 PTGS2 (0.44) PTGS2PTGS1HRH4
SCHEMBL5808581 0.83 PTGS2 (0.44) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL5558542 0.83 PTGS2 (0.57) CA1CA2PTGS2PTGS1HRH4
SCHEMBL5559101 0.83 PTGS2 (0.45) CA1CA2PTGS2PTGS1HRH4
SCHEMBL5554091 0.83 PTGS2 (0.57) CA1CA2PTGS2PTGS1HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed