SCHEMBL5554594

SCHEMBL5554594

CC(=O)Oc1c(C)n(C(=O)c2ccc(Br)cc2)c2cc(F)c(O)c(C)c12

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SRC P12931 4/20 0.36
PRKACA P17612 4/20 0.36
PRKACG P22612 4/20 0.36
PRKACB P22694 4/20 0.36
ALDH1A1 P00352 3/20 0.35
HPGD P15428 2/20 0.35
PTGS2 P35354 4/20 0.32
AKR1C3 P42330 3/20 0.32
AKR1C2 P52895 3/20 0.32
MAPT P10636 4/20 0.31
TSHR P16473 1/20 0.31
KDM4E B2RXH2 2/20 0.30
GAA P10253 2/20 0.30
HTT P42858 2/20 0.30
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
KMT2A Q03164 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5554224 0.88 AKR1C3 (0.35) ALDH1A1HPGDPTGS2AKR1C3AKR1C2
SCHEMBL5558391 0.87 SRC (0.42) SRCPRKACAPRKACGPRKACBALDH1A1
SCHEMBL5797596 0.86 AKR1C3 (0.45) PTGS2AKR1C3AKR1C2MAPTTSHR
SCHEMBL5559390 0.81 AKR1C3 (0.42) PTGS2AKR1C3AKR1C2MAPTKDM4E
SCHEMBL5560536 0.79 KMT2A (0.36) PTGS2AKR1C3AKR1C2MEN1KMT2A
SCHEMBL5558850 0.79 AKR1C3 (0.40) PTGS2AKR1C3AKR1C2MAPTHTT
SCHEMBL5558223 0.78 PTGS2 (0.35) HPGDPTGS2AKR1C3AKR1C2
SCHEMBL5561193 0.77 HPGD (0.34) ALDH1A1HPGDPTGS2AKR1C3AKR1C2
SCHEMBL5554202 0.77 TACR3 (0.33) PTGS2AKR1C3AKR1C2
SCHEMBL5560242 0.77 PPARG (0.37) PTGS2AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed