SCHEMBL5554700

SCHEMBL5554700

Cc1c(CC(=O)OC(=O)C(c2c(C)n(C(=O)c3ccc(Cl)cc3)c3cc(F)c(O)cc23)C(C)C)c2cc(O)c(F)cc2n1C(=O)c1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.49
AKR1C3 P42330 2/20 0.48
CNR2 P34972 1/20 0.48
AKR1C2 P52895 1/20 0.48
PTGS1 P23219 3/20 0.47
HTR1A P08908 1/20 0.47
PKM P14618 1/20 0.47
GLO1 Q04760 1/20 0.47
HIF1A Q16665 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5554698 0.86 PTGS2 (0.55) PTGS2AKR1C3AKR1C2PTGS1HTR1A
SCHEMBL5554695 0.86 AKR1C3 (0.59) PTGS2AKR1C3AKR1C2PTGS1GLO1
SCHEMBL6423743 0.83 PTGS2 (0.46) PTGS2AKR1C3AKR1C2PTGS1GLO1
SCHEMBL5814349 0.80 PTGS2 (0.45) PTGS2AKR1C3AKR1C2PTGS1
SCHEMBL5814350 0.80 PTGS2 (0.45) PTGS2AKR1C3AKR1C2PTGS1
SCHEMBL2000986 0.80 AKR1C3 (0.72) PTGS2AKR1C3AKR1C2PTGS1HTR1A
SCHEMBL5797344 0.80 PTGS2 (0.53) PTGS2AKR1C3AKR1C2PTGS1HTR1A
SCHEMBL5800814 0.79 AKR1C3 (0.48) PTGS2AKR1C3AKR1C2PTGS1GLO1
SCHEMBL5558176 0.79 PTGS2 (0.64) PTGS2AKR1C3CNR2AKR1C2PTGS1
SCHEMBL5559410 0.78 PTGS2 (0.58) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed