SCHEMBL5554900

SCHEMBL5554900

CCc1[nH]c(-c2cccc3ccccc23)nc1C(=O)N1CCN(C2CCC2)CC1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 6/20 0.43
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HIF1A Q16665 1/20 0.41
ACACB O00763 4/20 0.40
ACACA Q13085 4/20 0.40
HRH3 Q9Y5N1 3/20 0.40
SPR P35270 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3400872 0.81 LMNA (0.46) HTR2CKDM4EALDH1A1MEN1KMT2A
SCHEMBL13072005 0.81 KDM4E (0.43) KDM4EALDH1A1MEN1KMT2AHIF1A
SCHEMBL14545934 0.80 KDM4E (0.43) KDM4EALDH1A1MEN1KMT2AHIF1A
SCHEMBL3405422 0.79 LMNA (0.48) HTR2CKDM4EALDH1A1MEN1KMT2A
SCHEMBL14545939 0.78 ACACB (0.44) HTR2CKDM4EALDH1A1MEN1KMT2A
SCHEMBL5549726 0.78 GAA (0.35) HTR2CKDM4EALDH1A1
SCHEMBL3401298 0.78 HTR2C (0.46) HTR2CKDM4EALDH1A1MEN1KMT2A
SCHEMBL14546059 0.77 HRH3 (0.46) HTR2CKDM4EALDH1A1MEN1KMT2A
SCHEMBL3405430 0.76 ACACB (0.47) KDM4EALDH1A1MEN1KMT2AHIF1A
SCHEMBL3401027 0.76 HTR2C (0.46) HTR2CKDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1848428-A2 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORPORATION (US) 2007-10-31 EP disclosed
WO-2006089076-A2 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORPORATION (US) 2006-08-24 WO disclosed