SCHEMBL5558060

SCHEMBL5558060

O=C(CCCl)N1C(=O)CCC1=O

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.38
NPC1 O15118 1/20 0.32
MITF O75030 1/20 0.32
RAB9A P51151 1/20 0.32
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5559964 0.87 LMNA (0.35) LMNANPC1MITFRAB9APOLB
SCHEMBL5557939 0.85 LMNA (0.34) LMNANPC1MITFRAB9APOLB
SCHEMBL5558055 0.81 NPC1 (0.47) LMNANPC1MITFRAB9APOLB
SCHEMBL29366012 0.81 LMNA (0.40) LMNAPOLB
SCHEMBL16203504 0.79 LMNA (0.39) LMNAPOLB
SCHEMBL31733909 0.79 LMNA (0.39) LMNAPOLB
SCHEMBL12337488 0.77 LMNA (0.48) LMNAPOLB
SCHEMBL16135507 0.77 LMNA (0.38) LMNAPOLB
SCHEMBL8178094 0.77 CES1 (0.43) LMNAPOLB
SCHEMBL8649771 0.77 LMNA (0.38) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7220746-B2 Pyrrolidinedione substituted piperidine-phthalazones as PDE4 inhibitors ALTANA PHARMA AG (DE) 2007-05-22 US disclosed
EP-1537100-B1 PYRROLIDINEDIONE SUBSTITUTED PIPERIDINE-PHTHALAZONES AS PDE4 INHIBITORS ALTANA PHARMA AG (DE) 2007-04-25 EP disclosed
US-20060160813-A1 Pyrrolidinedione substituted piperidine-phtalazones as pde4 inhibitors ALTANA PHARMA AG (DE) 2006-07-20 US disclosed
EP-1537100-A1 PYRROLIDINEDIONE SUBSTITUTED PIPERIDINE-PHTHALAZONES AS PDE4 INHIBITORS ALTANA Pharma AG (DE) 2005-06-08 EP disclosed
WO-2004018457-A1 PYRROLIDINEDIONE SUBSTITUTED PIPERIDINE-PHTHALAZONES AS PDE4 INHIBITORS ALTANA PHARMA AG (DE) 2004-03-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060160813-A1 Pyrrolidinedione substituted piperidine-phtalazones as pde4 inhibitors PDE4A, PDE4B, PDE3B LMNA 3936/4885NPC1 4373/4885MITF 3716/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.