SCHEMBL5558368

SCHEMBL5558368

CC(C)CN[C@@H]1CC[C@H](N2CCC(Nc3ccccc3C(F)(F)F)C2=O)[C@H](CS(=O)(=O)c2ccccc2)C1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 20/20 0.52
KCNH2 Q12809 4/20 0.52
CCR5 P51681 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4417562 0.86 CCR2 (0.69) CCR2KCNH2CCR5
SCHEMBL4417558 0.86 CCR2 (0.69) CCR2KCNH2CCR5
Trifluoroacetic Acid SCHEMBL5558145 0.86 CCR2 (0.49) CCR2KCNH2CCR5
Trifluoroacetic Acid SCHEMBL5558180 0.84 CCR2 (0.57) CCR2KCNH2CCR5
Trifluoroacetic Acid SCHEMBL5027367 0.83 CCR2 (0.69) CCR2KCNH2CCR5
SCHEMBL5029327 0.80 CCR2 (0.49) CCR2KCNH2
SCHEMBL4414970 0.80 CCR2 (0.49) CCR2KCNH2
Trifluoroacetic Acid SCHEMBL5554138 0.80 CCR2 (0.51) CCR2KCNH2CCR5
SCHEMBL4416862 0.78 CCR2 (0.64) CCR2KCNH2CCR5
SCHEMBL4423062 0.77 CCR2 (0.45) CCR2KCNH2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1606255-A4 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2007-02-07 EP claimed
EP-1606255-A2 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Bristol-Myers Squibb Company (US) 2005-12-21 EP claimed
WO-2004071460-A2 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2004-08-26 WO claimed