SCHEMBL5559104

SCHEMBL5559104

Cc1c(CC=O)c2cc(O)ccc2n1C(=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.58
PTGS1 P23219 7/20 0.58
AKR1C3 P42330 6/20 0.44
AKR1C2 P52895 5/20 0.44
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
PTGES O14684 1/20 0.43
ABCC3 O15438 1/20 0.43
ABCC4 O15439 1/20 0.43
ABCB11 O95342 1/20 0.43
MT-CO2 P00403 1/20 0.43
LMNA P02545 1/20 0.43
ALB P02768 1/20 0.43
CYP1A2 P05177 1/20 0.43
ABCB1 P08183 1/20 0.43
ALOX5 P09917 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
CXCL8 P10145 1/20 0.43
AR P10275 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12628273 0.89 PTGS2 (0.73) PTGS2PTGS1AKR1C3AKR1C2KDM4E
SCHEMBL2002967 0.85 PTGS1 (0.79) PTGS2PTGS1AKR1C3AKR1C2KDM4E
SCHEMBL5558945 0.84 PTGS2 (0.58) PTGS2PTGS1AKR1C3AKR1C2KDM4E
SCHEMBL5808388 0.84 PTGS2 (0.55) PTGS2PTGS1AKR1C3AKR1C2KDM4E
SCHEMBL6425344 0.84 PTGS2 (0.64) PTGS2PTGS1AKR1C3AKR1C2KDM4E
SCHEMBL5559534 0.83 PTGS2 (0.64) PTGS2PTGS1TRPV1
SCHEMBL6423952 0.83 PTGS2 (0.62) PTGS2PTGS1AKR1C3AKR1C2MAPT
SCHEMBL6466294 0.81 PTGS2 (0.63) PTGS2PTGS1AKR1C3AKR1C2KDM4E
SCHEMBL5558489 0.81 PTGS2 (0.73) PTGS2PTGS1TRPV1
SCHEMBL5553933 0.81 PTGS2 (0.67) PTGS2PTGS1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed