SCHEMBL5559366

SCHEMBL5559366

CCOC(=O)ON1CCC2(CC1)CCn1c(nc(-c3ccncn3)cc1=O)N2CC(=O)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.41
CYP2D6 P10635 4/20 0.36
CYP1A2 P05177 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5554750 0.96 GSK3B (0.40) GSK3BCYP2D6CYP1A2
SCHEMBL5560969 0.90 GSK3B (0.41) GSK3BCYP2D6CYP1A2
SCHEMBL4418104 0.90 GSK3B (0.44) GSK3BCYP2D6CYP1A2
SCHEMBL5559159 0.89 GSK3B (0.40) GSK3BCYP2D6CYP1A2
SCHEMBL5564271 0.88 GSK3B (0.42) GSK3BCYP2D6CYP1A2
SCHEMBL4552623 0.87 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL5554252 0.87 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL5554665 0.86 GSK3B (0.48) GSK3BCYP2D6CYP1A2
SCHEMBL3367128 0.86 GSK3B (0.45) GSK3BCYP2D6CYP1A2
SCHEMBL3366553 0.86 GSK3B (0.45) GSK3BCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1699795-B1 SUBSTITUTED 8'-PYRI(MI)DINYL-DIHYDROSPIRO-[CYCLOALKLYMINE]-PYRIMIDO[1,2A]PYRIMIDIN-6-ONE DERIVATIVES SANOFI AVENTIS (FR) 2007-04-25 EP claimed