SCHEMBL5559159

SCHEMBL5559159

CCOC(=O)ON1CCC2(CC1)CCn1c(nc(-c3ccncn3)cc1=O)N2C[C@@H](O)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 19/20 0.40
CYP2D6 P10635 5/20 0.38
CYP1A2 P05177 2/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5554219 0.96 GSK3B (0.39) GSK3BCYP2D6CYP1A2KDM4EALDH1A1
SCHEMBL5559518 0.90 GSK3B (0.43) GSK3BCYP2D6CYP1A2KDM4EALDH1A1
SCHEMBL4431426 0.90 KDM4E (0.45) GSK3BCYP2D6CYP1A2KDM4EALDH1A1
SCHEMBL5559366 0.89 GSK3B (0.41) GSK3BCYP2D6CYP1A2
SCHEMBL5563111 0.88 GSK3B (0.42) GSK3BCYP2D6CYP1A2KDM4EALDH1A1
SCHEMBL5560982 0.87 GSK3B (0.42) GSK3BCYP2D6CYP1A2KDM4EALDH1A1
SCHEMBL5559918 0.87 GSK3B (0.42) GSK3BCYP2D6CYP1A2KDM4EALDH1A1
SCHEMBL5560979 0.87 GSK3B (0.42) GSK3BCYP2D6CYP1A2KDM4EALDH1A1
SCHEMBL4431960 0.87 GSK3B (0.42) GSK3BCYP2D6CYP1A2KDM4EALDH1A1
SCHEMBL5554765 0.86 GSK3B (0.42) GSK3BCYP2D6CYP1A2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1699795-B1 SUBSTITUTED 8'-PYRI(MI)DINYL-DIHYDROSPIRO-[CYCLOALKLYMINE]-PYRIMIDO[1,2A]PYRIMIDIN-6-ONE DERIVATIVES SANOFI AVENTIS (FR) 2007-04-25 EP claimed