SCHEMBL5559490

SCHEMBL5559490

O=C(CN1c2nc(-c3ccncc3)cc(=O)n2CCC12CCN(C(=O)C1CC1)CC2)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.41
ACACB O00763 6/20 0.38
ACACA Q13085 6/20 0.38
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
VCP P55072 1/20 0.36
ALDH1A1 P00352 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
GRM5 P41594 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4420489 0.97 GSK3B (0.40) GSK3BACACBACACAITGB3ITGA2B
SCHEMBL4420806 0.96 ACACB (0.42) GSK3BACACBACACAALDH1A1KDM4E
SCHEMBL4422560 0.95 GSK3B (0.40) GSK3BACACBACACAITGB3ITGA2B
SCHEMBL4424995 0.92 GSK3B (0.39) GSK3BACACBACACAITGB3ITGA2B
SCHEMBL4424997 0.91 ACACB (0.39) GSK3BACACBACACAITGB3ITGA2B
SCHEMBL5554395 0.90 GSK3B (0.44) GSK3BALDH1A1CYP1A2CYP2D6TSHR
SCHEMBL3366965 0.90 GSK3B (0.47) GSK3BALDH1A1CYP1A2CYP2D6TSHR
SCHEMBL3368275 0.89 GSK3B (0.46) GSK3BALDH1A1CYP1A2CYP2D6TSHR
SCHEMBL3364367 0.89 GSK3B (0.46) GSK3BALDH1A1CYP1A2CYP2D6TSHR
SCHEMBL5554655 0.87 GSK3B (0.43) GSK3BACACBACACAITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1699795-B1 SUBSTITUTED 8'-PYRI(MI)DINYL-DIHYDROSPIRO-[CYCLOALKLYMINE]-PYRIMIDO[1,2A]PYRIMIDIN-6-ONE DERIVATIVES SANOFI AVENTIS (FR) 2007-04-25 EP claimed
EP-1699795-B1 SUBSTITUTED 8'-PYRI(MI)DINYL-DIHYDROSPIRO-[CYCLOALKLYMINE]-PYRIMIDO[1,2A]PYRIMIDIN-6-ONE DERIVATIVES SANOFI AVENTIS (FR) 2007-04-25 EP disclosed