SCHEMBL4424997

SCHEMBL4424997

O=C(CN1c2nc(-c3ccncc3)cc(=O)n2CCC12CCN(C(=O)C1CCCCC1)C2)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.39
ACACA Q13085 2/20 0.39
GSK3B P49841 3/20 0.39
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
USP19 O94966 4/20 0.36
CYP2C9 P11712 1/20 0.35
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
ITGB3 P05106 2/20 0.34
ITGA2B P08514 2/20 0.34
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4424995 0.98 GSK3B (0.39) ACACBACACAGSK3BKDM4EMEN1
SCHEMBL4422560 0.96 GSK3B (0.40) ACACBACACAGSK3BKDM4EMEN1
SCHEMBL4420806 0.95 ACACB (0.42) ACACBACACAGSK3BKDM4EMEN1
SCHEMBL4420489 0.93 GSK3B (0.40) ACACBACACAGSK3BKDM4EMEN1
SCHEMBL5559490 0.91 GSK3B (0.41) ACACBACACAGSK3BKDM4EMEN1
SCHEMBL4425247 0.90 GSK3B (0.42) GSK3BKDM4EMEN1ALDH1A1HPGD
SCHEMBL4432305 0.89 GSK3B (0.43) GSK3BALDH1A1USP19CYP2C9
SCHEMBL4421963 0.88 GSK3B (0.40) ACACBACACAGSK3BUSP19CYP2C9
SCHEMBL4421961 0.88 GSK3B (0.40) ACACBACACAGSK3BUSP19CYP2C9
SCHEMBL4418561 0.88 GSK3B (0.42) GSK3BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1699795-B1 SUBSTITUTED 8'-PYRI(MI)DINYL-DIHYDROSPIRO-[CYCLOALKLYMINE]-PYRIMIDO[1,2A]PYRIMIDIN-6-ONE DERIVATIVES SANOFI AVENTIS (FR) 2007-04-25 EP claimed
US-7547705-B2 Substituted 8′-pyri(MI)dinyl-dihydrospiro-[cycloalkylamine]-pyrimido[1,2-a]pyrimidin-6-one derivatives SANOFI-AVENTIS (FR) 2009-06-16 US disclosed