SCHEMBL5559624

SCHEMBL5559624

O=C(c1cc(C(F)(F)F)cc(C(F)(F)F)c1)N1CCC2(CC1)C(=O)NCN2C(I)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 0.51
TSHR P16473 6/20 0.51
USP2 O75604 10/20 0.50
HSD17B10 Q99714 3/20 0.50
CYP2C9 P11712 6/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HIF1A Q16665 3/20 0.46
CYP2D6 P10635 3/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.46
TACR1 P25103 1/20 0.45
CYP1A2 P05177 4/20 0.45
CYP2C19 P33261 2/20 0.45
OPRD1 P41143 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5553371 0.81 CYP3A4 (0.61) CYP3A4TSHRUSP2HSD17B10CYP2C9
SCHEMBL5557693 0.81 CYP3A4 (0.55) CYP3A4TSHRUSP2HSD17B10CYP2C9
SCHEMBL5553322 0.78 USP2 (0.63) CYP3A4TSHRUSP2HSD17B10CYP2C9
SCHEMBL5558262 0.76 USP2 (0.49) CYP3A4TSHRUSP2HSD17B10CYP2C9
SCHEMBL5557778 0.76 CYP3A4 (0.49) CYP3A4TSHRUSP2HSD17B10CYP2C9
SCHEMBL5557913 0.76 PLD2 (0.55) CYP3A4TSHRUSP2HSD17B10HIF1A
SCHEMBL5553130 0.74 CYP3A4 (0.64) CYP3A4TSHRUSP2HSD17B10CYP2C9
SCHEMBL5557707 0.74 USP2 (0.53) CYP3A4TSHRUSP2HSD17B10CYP2C9
SCHEMBL5557466 0.74 USP2 (0.55) CYP3A4TSHRUSP2HSD17B10CYP2C9
SCHEMBL5557537 0.74 USP2 (0.52) CYP3A4TSHRUSP2HSD17B10CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1292596-B1 1,3,8-TRIAZA-SPIRO¬4,5 DECAN-4-ONE DERIVATIVES AS NEUROKININ RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2007-12-19 EP disclosed