SCHEMBL5559822

SCHEMBL5559822

Cc1c(CC=O)c2c(F)c(O)c(F)cc2n1C(=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.38
AKR1C2 P52895 3/20 0.38
PTGS2 P35354 7/20 0.36
PTGS1 P23219 5/20 0.36
HPGD P15428 1/20 0.34
ABCB1 P08183 2/20 0.34
TSHR P16473 1/20 0.33
ALOX5 P09917 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5558932 0.89 AKR1C3 (0.39) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL5808070 0.89 AKR1C3 (0.48) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL5553916 0.88 AKR1C3 (0.40) AKR1C3AKR1C2PTGS2PTGS1HPGD
SCHEMBL5553862 0.87 AKR1C3 (0.51) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL5814553 0.87 CNR1 (0.40) AKR1C3AKR1C2PTGS2PTGS1HPGD
SCHEMBL6423473 0.86 PTGS2 (0.45) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL5558650 0.85 PTGS2 (0.42) AKR1C3AKR1C2PTGS2PTGS1
SCHEMBL5559282 0.83 PTGS2 (0.42) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL5553794 0.83 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL5554132 0.83 PTGS2 (0.50) PTGS2PTGS1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed