SCHEMBL5560596

SCHEMBL5560596

COc1ccc(CCNC2CC2)cc1

nearest known ligand 0.76

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.65
KMT2A Q03164 1/20 0.65
KDM4E B2RXH2 2/20 0.57
SMN1; SMN2 Q16637 3/20 0.51
HTT P42858 1/20 0.50
MAPT P10636 1/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA5A P35218 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
GRIN1 Q05586 1/20 0.50
GRIN2B Q13224 1/20 0.50
HRH3 Q9Y5N1 2/20 0.49
LMNA P02545 1/20 0.49
ALDH1A1 P00352 1/20 0.49
TAAR1 Q96RJ0 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL787034 0.93 KDM4E (0.67) POLBKMT2AKDM4EHRH3ALDH1A1
SCHEMBL3692058 0.92 KMT2A (0.58) POLBKMT2AKDM4ESMN1; SMN2GRIN1
SCHEMBL3692055 0.92 KMT2A (0.58) POLBKMT2AKDM4ESMN1; SMN2GRIN1
SCHEMBL5561766 0.92 KDM4E (0.65) POLBKMT2AKDM4ESMN1; SMN2HTT
SCHEMBL14885856 0.89 POLB (0.58) POLBKMT2AKDM4ESMN1; SMN2HTT
SCHEMBL9995215 0.88 KMT2A (0.60) POLBKMT2AKDM4ESMN1; SMN2HRH3
SCHEMBL6483020 0.85 KMT2A (0.51) POLBKMT2AKDM4ESMN1; SMN2MAPT
SCHEMBL6496123 0.85 KMT2A (0.51) POLBKMT2AKDM4ESMN1; SMN2MAPT
SCHEMBL6483016 0.85 KMT2A (0.51) POLBKMT2AKDM4ESMN1; SMN2MAPT
SCHEMBL7026318 0.83 KMT2A (0.55) POLBKMT2AKDM4ESMN1; SMN2GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761509-A2 SUBSTITUTED CYCLOALKYL DERIVATIVES FOR THE TREATMENT OF RESPIRATORY DISEASES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-03-14 EP disclosed
WO-2005111002-A2 SUBSTITUTED CYCLOALKYL DERIVATIVES FOR USE IN THE TREATMENT OF RESPIRATORY DISEASES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-24 WO disclosed