SCHEMBL5560833

SCHEMBL5560833

Cc1c(C[C]=O)c2cc(O)c(Cl)cc2n1C(=O)c1ccc(OC(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.44
PTGS1 P23219 5/20 0.44
PPARG P37231 2/20 0.43
AKR1C3 P42330 4/20 0.43
AKR1C2 P52895 3/20 0.43
ABCB1 P08183 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
PTGES O14684 1/20 0.43
ABCC3 O15438 1/20 0.43
ABCC4 O15439 1/20 0.43
ABCB11 O95342 1/20 0.43
MT-CO2 P00403 1/20 0.43
LMNA P02545 1/20 0.43
ALB P02768 1/20 0.43
CYP1A2 P05177 1/20 0.43
ALOX5 P09917 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
CXCL8 P10145 1/20 0.43
AR P10275 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5442566 0.87 PTGS1 (0.59) PTGS2PTGS1PPARGAKR1C3AKR1C2
SCHEMBL5554640 0.86 PTGS2 (0.58) PTGS2PTGS1PPARGAKR1C3AKR1C2
SCHEMBL5554579 0.86 PTGS2 (0.47) PTGS2PTGS1PPARGAKR1C3AKR1C2
SCHEMBL5558497 0.85 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL5554600 0.84 PTGS2 (0.53) PTGS2
SCHEMBL5813369 0.83 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL5554433 0.83 PTGS2 (0.63) PTGS2PTGS1
SCHEMBL5812740 0.82 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL5798265 0.82 PTGS2 (0.53) PTGS2PTGS1PPARGAKR1C3AKR1C2
SCHEMBL5559900 0.82 PTGS2 (0.54) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed