SCHEMBL5564105

SCHEMBL5564105

COc1cc2c(cc1OC)NCC2

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.49
TSHR P16473 1/20 0.49
CYP3A4 P08684 1/20 0.48
MAPT P10636 1/20 0.48
HTR2A P28223 4/20 0.47
HTR2C P28335 4/20 0.47
HTR2B P41595 4/20 0.47
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
KDM4E B2RXH2 1/20 0.40
CHRNA7 P36544 1/20 0.40
MAOB P27338 1/20 0.40
SLC6A4 P31645 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10912768 0.88 MAPT (0.45) MAOATSHRCYP3A4MAPTHTR2A
SCHEMBL19411037 0.87 HTR2A (0.40) MAOATSHRCYP3A4MAPTHTR2A
SCHEMBL12420344 0.86 HTR2A (0.43) MAOATSHRCYP3A4MAPTHTR2A
SCHEMBL30340758 0.86 MAPT (0.43) MAOATSHRCYP3A4MAPTHTR2A
SCHEMBL5468971 0.86 MAPT (0.43) MAOATSHRCYP3A4MAPTHTR2A
SCHEMBL13942395 0.86 HTR2A (0.43) MAOATSHRCYP3A4MAPTHTR2A
Hydrochloric Acid SCHEMBL7373928 0.86 MAPT (0.44) MAOATSHRCYP3A4MAPTHTR2A
SCHEMBL1701913 0.85 MAOA (0.54) MAOAMAPTALDH1A1DRD2DRD4
SCHEMBL22340168 0.85 HTR2C (0.53) MAOATSHRCYP3A4MAPTHTR2A
SCHEMBL5186942 0.85 MAOA (0.54) MAOAALDH1A1DRD2DRD4CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 104 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6828443-B1 Dyes and colorants HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 2004-12-07 US claimed
EP-0575604-B2 INDOLINE PRODUCTS, METHODS FOR PREPARING SAME, AND USE THEREOF IN COSMETICS OREAL (FR) 2003-03-26 EP claimed
US-5776497-A OXIDATIVE POLYMERIZATION OF INDOLINE FOR COSMETICS L'OREAL (FR) 1998-07-07 US claimed
EP-0544874-B1 METHOD FOR PREPARING SUBMICRON PARTICLES IN THE PRESENCE OF LIPID VESICLES, AND CORRESPONDING COMPOSITIONS OREAL (FR) 1998-04-08 EP claimed
US-5670099-A PREPARING A DISPERSION OF LIPIDIC VESICLES FROM ATLEAST ONE LIPID, AN AQUEOUS PHASE ENCAPSULATED IN VESICLE, DISSOLVING POLYMERIZABLE INDOLIC OR INDOLINIC MONOMER WITH A POLYMERIZATION AGENT, REACTS WITH MONOMER FORMS PARTICLES L'OREAL (FR) 1997-09-23 US claimed
US-5583234-A Indoline-based products, processes for preparing them and their use in cosmetics L'OREAL (FR) 1996-12-10 US claimed
EP-0575605-B1 MINERAL OR ORGANIC PARTICLE BASED PRODUCT COMPRISING AN INDOLINE PRODUCT OREAL (FR) 1996-11-27 EP claimed
US-5496543-A COSMETICS L'OREAL (FR) 1996-03-05 US claimed
EP-0575604-B1 INDOLINE PRODUCTS, METHODS FOR PREPARING SAME, AND USE THEREOF IN COSMETICS OREAL (FR) 1995-12-06 EP claimed
EP-0575604-A1 INDOLINE PRODUCTS, METHODS FOR PREPARING SAME, AND USE THEREOF IN COSMETICS. OREAL (FR) 1993-12-29 EP claimed
WO-1993013744-A1 INDOLINE PRODUCTS, METHODS FOR PREPARING SAME, AND USE THEREOF IN COSMETICS L'OREAL (FR) 1993-07-22 WO claimed
EP-0544874-A1 METHOD FOR PREPARING SUBMICRON PARTICLES IN THE PRESENCE OF LIPID VESICLES, AND CORRESPONDING COMPOSITIONS L'OREAL (FR) 1993-06-09 EP claimed
WO-1993000068-A1 METHOD FOR PREPARING SUBMICRON PARTICLES IN THE PRESENCE OF LIPID VESICLES, AND CORRESPONDING COMPOSITIONS L'OREAL (FR) 1993-01-07 WO claimed
EP-4581028-A1 INDOLINE DERIVATIVES AS SEROTONERGIC AGENTS USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO Mindset Pharma Inc. (CA) 2025-07-09 EP disclosed
CN-120040333-A Preparation method of 5, 6-dihydroxyindoline 北京成宇化工有限公司 2025-05-27 CN disclosed
CN-119118902-A Synthesis method of 5, 6-dimethoxy isoindoline hydrochloride 郑州药领医药科技有限公司 2024-12-13 CN disclosed
WO-1993000068-A1 METHOD FOR PREPARING SUBMICRON PARTICLES IN THE PRESENCE OF LIPID VESICLES, AND CORRESPONDING COMPOSITIONS L'OREAL (FR) 1993-01-07 WO disclosed
EP-0462857-A1 Dyeing composition containing 5-6 dihydroxyindolines and keratinous fibres dyeing process L'OREAL (FR) 1991-12-27 EP disclosed
WO-1991017739-A1 OXIDATION COLORANTS FOR KERATIN FIBRES HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1991-11-28 WO disclosed
US-4159271-A CYCLIZATION OF A 2-HALOGENOPHENETHYLAMINE IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 1979-06-26 US disclosed