SCHEMBL5564657

SCHEMBL5564657

CC(=NOCc1ccc(-c2ccccc2)cc1)c1ccc(CCC(N)(CO)CO)cc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 14/20 0.55
L3MBTL1 Q9Y468 2/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
S1PR3 Q99500 2/20 0.47
TNNC1 P63316 5/20 0.43
SGPL1 O95470 1/20 0.43
S1PR4 O95977 1/20 0.43
GPR183 P32249 1/20 0.43
CERS2 Q96G23 1/20 0.43
S1PR5 Q9H228 1/20 0.43
LMNA P02545 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11927165 1.00 S1PR1 (0.55) S1PR1L3MBTL1NPC1RAB9ASMN1; SMN2
SCHEMBL11927465 0.89 S1PR1 (0.67) S1PR1S1PR3S1PR4S1PR5
SCHEMBL5559723 0.89 S1PR1 (0.67) S1PR1S1PR3S1PR4S1PR5
SCHEMBL27625020 0.84 S1PR1 (0.44) S1PR1S1PR3TNNC1SGPL1S1PR4
SCHEMBL14593245 0.82 S1PR1 (0.51) S1PR1S1PR3TNNC1SGPL1S1PR4
SCHEMBL6529404 0.81 S1PR1 (0.59) S1PR1RAB9AS1PR3TNNC1SGPL1
SCHEMBL14593328 0.81 SMN1; SMN2 (0.43) S1PR1SMN1; SMN2S1PR3TNNC1SGPL1
SCHEMBL5397755 0.81 SMN1; SMN2 (0.43) S1PR1SMN1; SMN2S1PR3TNNC1SGPL1
SCHEMBL5566429 0.79 S1PR1 (0.59) S1PR1S1PR3S1PR4S1PR5
SCHEMBL27625019 0.78 S1PR1 (0.43) S1PR1S1PR3TNNC1SGPL1S1PR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1594508-B1 NOVEL BICYCLIC COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2012-08-08 EP disclosed
US-7256206-B2 1-[4-(3-Amino-4-hydroxy-3-hydroxymethyl-butyl)-phenyl]-ethanone-O-biphenyl-4-ylmethyl-oxime, used as modulators of lipid activated G-protein coupled receptors specific for sphingosine-1-phosphate; prevention of autoimmune diseases or as angiogenesis inhibitors IRM LLC (BM) 2007-08-14 US disclosed
US-20040248952-A1 Novel bicyclic compounds and compositions IRM LLC, A DELAWARE LIMITED LIABILITY COMPANY (BM) 2004-12-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040248952-A1 Novel bicyclic compounds and compositions S1PR1, S1PR3, S1PR5 S1PR1 1/4885L3MBTL1 3502/4885NPC1 567/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.