SCHEMBL5568600

SCHEMBL5568600

CC[C@H](N)C(=O)N1c2ccc(Cl)cc2C[C@@H]1OC(=O)NCCCl

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
CYP1A2 P05177 2/20 0.42
KDM4E B2RXH2 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CYP2C19 P33261 1/20 0.35
AADAT Q8N5Z0 1/20 0.33
SRD5A1 P18405 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6242182 0.91 KDM4E (0.52) ALDH1A1CYP1A2KDM4ECYP3A4CYP2D6
SCHEMBL5568426 0.87 KDM4E (0.39) ALDH1A1CYP1A2KDM4ECYP3A4CYP2D6
SCHEMBL5563144 0.83 KDM4E (0.61) ALDH1A1CYP1A2KDM4ECYP3A4CYP2D6
SCHEMBL6244677 0.83 KDM4E (0.53) ALDH1A1CYP1A2KDM4ECYP3A4CYP2D6
SCHEMBL6242771 0.79 KDM4E (0.60) ALDH1A1CYP1A2KDM4ECYP3A4CYP2D6
Trifluoroacetic Acid SCHEMBL5567550 0.78 KDM4E (0.55) ALDH1A1CYP1A2KDM4ECYP3A4CYP2D6
SCHEMBL6242475 0.77 KDM4E (0.70) ALDH1A1CYP1A2KDM4ECYP3A4CYP2D6
SCHEMBL6240896 0.77 KDM4E (0.57) ALDH1A1CYP1A2KDM4ECYP3A4CYP2D6
SCHEMBL6242776 0.77 KDM4E (0.60) ALDH1A1CYP1A2KDM4ECYP3A4CYP2D6
SCHEMBL5563867 0.76 KDM4E (0.54) ALDH1A1CYP1A2KDM4ECYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042288-B1 TRIPEPTIDYL PEPTIDASE INHIBITORS INST NAT SANTE RECH MED (FR) 2007-11-07 EP claimed