SCHEMBL5570765

SCHEMBL5570765

CC1CC(c2nc3ccccc3s2)C[N]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.54
MEN1 O00255 2/20 0.54
UBE2M P61081 7/20 0.43
DCUN1D1 Q96GG9 7/20 0.43
GAA P10253 2/20 0.43
ALDH1A1 P00352 5/20 0.43
TP53 P04637 3/20 0.43
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
GRM2 Q14416 1/20 0.43
PDE10A Q9Y233 1/20 0.42
LMNA P02545 4/20 0.41
ALOX12 P18054 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
RECQL P46063 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17058991 0.80 KMT2A (0.58) KMT2AMEN1UBE2MDCUN1D1GAA
SCHEMBL16545296 0.77 KMT2A (0.59) KMT2AMEN1UBE2MDCUN1D1GAA
SCHEMBL9533470 0.77 KMT2A (0.77) KMT2AMEN1UBE2MDCUN1D1GAA
SCHEMBL24819771 0.76 KMT2A (0.57) KMT2AMEN1UBE2MDCUN1D1GAA
SCHEMBL19781780 0.76 MEN1 (0.53) KMT2AMEN1UBE2MDCUN1D1GAA
SCHEMBL5637621 0.74 KMT2A (0.73) KMT2AMEN1UBE2MDCUN1D1GAA
SCHEMBL1744058 0.74 KMT2A (0.73) KMT2AMEN1UBE2MDCUN1D1GAA
SCHEMBL7963995 0.74 KMT2A (0.67) KMT2AMEN1UBE2MDCUN1D1GAA
SCHEMBL7964001 0.74 KMT2A (0.67) KMT2AMEN1UBE2MDCUN1D1GAA
SCHEMBL7963999 0.74 KMT2A (0.67) KMT2AMEN1UBE2MDCUN1D1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778639-A2 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR Technology, Inc. (US) 2007-05-02 EP claimed
WO-2006020049-A2 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR TECHNOLOGY, INC. (US) 2006-02-23 WO claimed
EP-1778639-A2 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR Technology, Inc. (US) 2007-05-02 EP disclosed
WO-2006020049-A2 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR TECHNOLOGY, INC. (US) 2006-02-23 WO disclosed