SCHEMBL5573121

SCHEMBL5573121

CCCN1Cc2ccccc2C1(OCCc1ccccn1)c1ccc(OCOCC[Si](C)(C)C)cc1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 5/20 0.47
TP53 P04637 4/20 0.47
HPGD P15428 2/20 0.31
MEN1 O00255 1/20 0.31
HSD17B10 Q99714 1/20 0.31
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4914752 0.81 MDM2 (0.74) MDM2TP53
SCHEMBL4914758 0.81 MDM2 (0.74) MDM2TP53
SCHEMBL8272068 0.81 MDM2 (0.59) MDM2TP53HPGDHSD17B10
SCHEMBL5573053 0.78 TP53 (0.46) MDM2TP53
SCHEMBL4914047 0.66 MDM2 (0.68) MDM2TP53
SCHEMBL4914049 0.66 MDM2 (0.68) MDM2TP53
SCHEMBL8272067 0.66 MDM2 (0.53) MDM2TP53
SCHEMBL4912863 0.64 MDM2 (1.00) MDM2TP53HSD17B10
SCHEMBL4912856 0.64 MDM2 (1.00) MDM2TP53HSD17B10
SCHEMBL4912554 0.63 MDM2 (0.65) MDM2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786773-A1 ISOINDOLIN-1-ONE DERIVATIVES Cancer Research Technology Limited (GB) 2007-05-23 EP disclosed
WO-2006024837-A1 ISOINDOLIN-1-ONE DERIVATIVES CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2006-03-09 WO disclosed