SCHEMBL5573053

SCHEMBL5573053

CCCN1Cc2ccccc2C1(OCc1cc(OC)c(O)c(OC)c1)c1ccc(OCOCC[Si](C)(C)C)cc1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TP53 P04637 6/20 0.46
MDM2 Q00987 6/20 0.46
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5570568 0.84 TP53 (0.62) TP53MDM2KDM4EGAAMAPT
SCHEMBL4913263 0.82 MDM2 (0.72) TP53MDM2
SCHEMBL4913256 0.82 MDM2 (0.72) TP53MDM2
SCHEMBL5573121 0.78 MDM2 (0.47) TP53MDM2
SCHEMBL4916051 0.76 MDM2 (0.73) TP53MDM2
SCHEMBL4916054 0.76 MDM2 (0.73) TP53MDM2
SCHEMBL12017330 0.66 MDM2 (0.51) TP53MDM2
SCHEMBL12017329 0.66 MDM2 (0.51) TP53MDM2
SCHEMBL4911242 0.66 TP53 (0.68) TP53MDM2
SCHEMBL8272070 0.66 MDM2 (0.57) TP53MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786773-A1 ISOINDOLIN-1-ONE DERIVATIVES Cancer Research Technology Limited (GB) 2007-05-23 EP disclosed
WO-2006024837-A1 ISOINDOLIN-1-ONE DERIVATIVES CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2006-03-09 WO disclosed